Position: Post-Doc
Email: alessio.nocentini@unifi.it
Phone: +39 055 4573685
Location: Firenze
Medicinal Chemistry Drug Design Organic Chemistry, Molecular Modelling, Enzymology
Docente di Analisi dei Medicinali I – modulo II B030128 (B054) CdLM in Farmacia, Scuola di Scienze della salute umana
2014–2017 PhD cum laude in Area del Farmaco e Trattamenti Innovativi: Curriculum Scienze Farmaceutiche (Medicinal Chemistry), NEUROFARBA Department, University of Florence - PhD Supervisor: Prof. Paola Gratteri 2008–2014 MSc, 110/110 cum laude in Pharmaceutical Chemistry and Technology, Pharmacy, University of Florence CURRENT AND PREVIOUS POSITION 2023–present RTD-b (Assistant Professor, SSD CHIM/08), NEUROFARBA Department, University of Florence, Italy 2020–2023 RTD-a (Assistant Professor, SSD CHIM/08), NEUROFARBA Department, University of Florence, Italy 2017–2020 Postdoctoral research fellowships, Supervisor: Prof. Claudiu T. Supuran, Prof. Paola Gratteri, NEUROFARBA Department, University of Florence
Premio Miglior Tesi di Dottorato 2018, Divisione di Chimica Farmaceutica, Società Chimica Italiana
Therapeutic Applications of Carbonic Anhydrase Inhibitors in Ophthalmology
- Giovannuzzi S. - Nocentini Alessio - Supuran C.T.Mechanisms of Carbonic Anhydrase Catalysis and Inhibition
- Raghav N. - Supuran C.T. - Nocentini AlessioApplications of Carbonic Anhydrase Inhibitors in Arthritis, Neuropathic Pain, Acute Mountain Sickness, and Cerebral Ischemia
- Nocentini Alessio - Pundeer R. - Supuran C.T.Bacterial Carbonic Anhydrase Inhibitor CAI0019 Demonstrates Efficacy in Enterococcus faecium Septicemic Peritonitis Mouse Model While Sparing the Microbiome
- Abutaleb N.S. - Holly K.J. - Metcalfe C.K. - Abouelkhair A.A. - Tharra P.R. - Shrinidhi A. - Abdelsattar A.S. - Burgo V. - Melotte G. - Akin-Olabiyi T. - Knoblauch S. - Ramaswamy R. - Woodson C. - Thirumalaikumar V.P. - Rodriguez J.A. - Yeo F.J. - Snell O.C. - Nocentini Alessio - Sundararajan A. - Olson M.R. - Supuran C.T. - Seleem M.N. - Flaherty D.P.Discovery of enaminone-linked benzofuran derivatives as dual VEGFR-2/hCA IX inhibitors exhibiting hypoxia-mediated chemosensitization
- Eldehna W.M. - Elsayed Z.M. - Elnagar M.R. - Ammara A. - Elkotamy M.S. - Monir R. - Nocentini Alessio - Al-Sanea M.M. - Supuran C.T. - Tawfik H.O. - Abdel-Aziz H.A. - Negmeldin A.T.First-in-Class Dual PDGFR/Carbonic Anhydrase IX/XII Inhibitors: 6,7-Dimethoxyquinoline-Sulfonamides as Promising Antileukemic Agents
- Roshdy E. - Řezníčková E. - Elbadawi M.M. - Celik I. - Giovannuzzi S. - Veselá D. - Vojáčková V. - Krňávková P. - Nocentini Alessio - Supuran C.T. - Kryštof V. - Eldehna W.M. - Abe M.Targeting Metabolic and pH Regulatory Pathways in Cancer via Dual Inhibition of Nicotinamide Phosphoribosyltransferase and Carbonic Anhydrases IX and XII
- Paoletti N. - Giovannuzzi S. - Gasparrini M. - Ammara A. - Zaroon Z. - Raffaelli N. - De Nigris F. - Gratteri P. - Supuran C.T. - Nocentini Alessio4-(5-Chloro-3-(3,4,5-trimethoxybenzoyl)-1H-indol-1-yl)benzenesulfonamide: A Novel Polypharmacology Agent to Target Carbonic Anhydrase IX and XII With Improved Selectivity, Wnt/β-Catenin Signaling Pathway, and P-Glycoprotein
- Puxeddu M. - Bordone R. - Colla C. - Rotili G. - Coluccia A. - Sciò P. - Cuřínová P. - Nocentini Alessio - Supuran C.T. - Filiberti S. - Turati M. - Ronca R. - Kopecka J. - Riganti C. - Jimenez L. - Link W. - Bigogno C. - Dondio G. - Barba M. - Canettieri G. - Silvestri R. - La Regina G.Trypanosoma cruzi carbonic anhydrase inhibitors as a potential antiparasitic agent
- Lanera S.d.C. - Lara L.d.S. - Orlando L.M.R. - de Souza T.P. - de Oliveira E.C. - Paes V.B. - Figueiredo N.d.S. - Giovannuzzi S. - Nikitjuka A. - Nocentini Alessio - Winum J.Y. - Cardoso V.d.S. - Dias E.P.d.S. - Vermelho A.B. - Supuran C.T. - Pereira M.C.d.S.Consorzio interuniversitario per lo sviluppo dei Sistemi a Grande Interfase
Department of Chemistry, University of Florence - Via della Lastruccia 3 50019 - Sesto Fiorentino (FI)
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