Consorzio Interuniversitario per lo sviluppo dei Sistemi a Grande Interfase
Center for Colloid and Surface Science

Personal information

Position: Post-Doc

Email: alessio.nocentini@unifi.it

Phone: +39 055 4573685

Location: Firenze


Fields of Interest and Expertise

Medicinal Chemistry Drug Design Organic Chemistry, Molecular Modelling, Enzymology

Teaching

Docente di Analisi dei Medicinali I – modulo II B030128 (B054) CdLM in Farmacia, Scuola di Scienze della salute umana

Curriculum Vitae

2014–2017 PhD cum laude in Area del Farmaco e Trattamenti Innovativi: Curriculum Scienze Farmaceutiche (Medicinal Chemistry), NEUROFARBA Department, University of Florence - PhD Supervisor: Prof. Paola Gratteri 2008–2014 MSc, 110/110 cum laude in Pharmaceutical Chemistry and Technology, Pharmacy, University of Florence CURRENT AND PREVIOUS POSITION 2023–present RTD-b (Assistant Professor, SSD CHIM/08), NEUROFARBA Department, University of Florence, Italy 2020–2023 RTD-a (Assistant Professor, SSD CHIM/08), NEUROFARBA Department, University of Florence, Italy 2017–2020 Postdoctoral research fellowships, Supervisor: Prof. Claudiu T. Supuran, Prof. Paola Gratteri, NEUROFARBA Department, University of Florence

Awards

Premio Miglior Tesi di Dottorato 2018, Divisione di Chimica Farmaceutica, Società Chimica Italiana

Unit

Publications

Mechanisms of Carbonic Anhydrase Catalysis and Inhibition

- Raghav N. - Supuran C.T. - Nocentini Alessio
Subcellular Biochemistry

Bacterial Carbonic Anhydrase Inhibitor CAI0019 Demonstrates Efficacy in Enterococcus faecium Septicemic Peritonitis Mouse Model While Sparing the Microbiome

- Abutaleb N.S. - Holly K.J. - Metcalfe C.K. - Abouelkhair A.A. - Tharra P.R. - Shrinidhi A. - Abdelsattar A.S. - Burgo V. - Melotte G. - Akin-Olabiyi T. - Knoblauch S. - Ramaswamy R. - Woodson C. - Thirumalaikumar V.P. - Rodriguez J.A. - Yeo F.J. - Snell O.C. - Nocentini Alessio - Sundararajan A. - Olson M.R. - Supuran C.T. - Seleem M.N. - Flaherty D.P.
ACS Infectious Diseases

Discovery of enaminone-linked benzofuran derivatives as dual VEGFR-2/hCA IX inhibitors exhibiting hypoxia-mediated chemosensitization

- Eldehna W.M. - Elsayed Z.M. - Elnagar M.R. - Ammara A. - Elkotamy M.S. - Monir R. - Nocentini Alessio - Al-Sanea M.M. - Supuran C.T. - Tawfik H.O. - Abdel-Aziz H.A. - Negmeldin A.T.
Rsc Medicinal Chemistry

First-in-Class Dual PDGFR/Carbonic Anhydrase IX/XII Inhibitors: 6,7-Dimethoxyquinoline-Sulfonamides as Promising Antileukemic Agents

- Roshdy E. - Řezníčková E. - Elbadawi M.M. - Celik I. - Giovannuzzi S. - Veselá D. - Vojáčková V. - Krňávková P. - Nocentini Alessio - Supuran C.T. - Kryštof V. - Eldehna W.M. - Abe M.
Journal of Medicinal Chemistry

Targeting Metabolic and pH Regulatory Pathways in Cancer via Dual Inhibition of Nicotinamide Phosphoribosyltransferase and Carbonic Anhydrases IX and XII

- Paoletti N. - Giovannuzzi S. - Gasparrini M. - Ammara A. - Zaroon Z. - Raffaelli N. - De Nigris F. - Gratteri P. - Supuran C.T. - Nocentini Alessio
Journal of Medicinal Chemistry

4-(5-Chloro-3-(3,4,5-trimethoxybenzoyl)-1H-indol-1-yl)benzenesulfonamide: A Novel Polypharmacology Agent to Target Carbonic Anhydrase IX and XII With Improved Selectivity, Wnt/β-Catenin Signaling Pathway, and P-Glycoprotein

- Puxeddu M. - Bordone R. - Colla C. - Rotili G. - Coluccia A. - Sciò P. - Cuřínová P. - Nocentini Alessio - Supuran C.T. - Filiberti S. - Turati M. - Ronca R. - Kopecka J. - Riganti C. - Jimenez L. - Link W. - Bigogno C. - Dondio G. - Barba M. - Canettieri G. - Silvestri R. - La Regina G.
Chemmedchem

Trypanosoma cruzi carbonic anhydrase inhibitors as a potential antiparasitic agent

- Lanera S.d.C. - Lara L.d.S. - Orlando L.M.R. - de Souza T.P. - de Oliveira E.C. - Paes V.B. - Figueiredo N.d.S. - Giovannuzzi S. - Nikitjuka A. - Nocentini Alessio - Winum J.Y. - Cardoso V.d.S. - Dias E.P.d.S. - Vermelho A.B. - Supuran C.T. - Pereira M.C.d.S.
International Journal of Biological Macromolecules

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